2893. Denileukin Diftitox

Nomenclature

CAS number: 173146-27-5
N-l-Methionyl-387-l-histidine-388-l-alanine-1-388-toxin (Corynebacterium diphtheriae strain C7) (388→2′)-protein with 2-133-interleukin 2 (human clone pTIL2-21a); DAB389IL2; LY-335348; Ontak (Ligand).

Description and references

Recombinant fusion protein consisting of the catalytic and translocation domains of diphtheria toxin fused to interleukin 2, q.v. Immunotoxin that selectively targets eukaryotic cells expressing the interleukin 2 receptor. Prepn: D. Williams et al., J. Biol. Chem. 265, 11885 (1990). Clinical evaluation in cutaneous T cell lymphoma: M. Duvic et al., Am. J. Hematol. 58, 87 (1998). Review of development and clinical experience: F. M. Foss et al., Curr. Top. Microbiol. Immunol. 234, 63-81 (1998).

Therapeutic Category

Antineoplastic.

Keywords

Antineoplastic; Immunotoxins