3506. Eculizumab

Nomenclature

CAS number: 219685-50-4
Anti-(human complement C5 α-chain)(human-mouse monoclonal 5G1.1 heavy chain)immunoglobulin, disulfide with human-mouse monoclonal 5G1.1 light chain, dimer; h5G1.1 Fab; h5G1.1VHC + h5G1.1VLC; Soliris (Alexion).

Description and references

Humanized monoclonal antibody directed against complement component C5; designed to prevent activation of complement-mediated inflammation and tissue injury. Prepn: M. J. Evans et al., WO 9529697; eidem, US 6355245 (1995, 2002 both to Alexion); and complement inhibition study: T. C. Thomas et al., Mol. Immunol. 33, 1389 (1996). Overview of development and therapeutic potential: M. Kaplan, Curr. Opin. Investig. Drugs 3, 1017-1023 (2002). Clinical trial in paroxysmal nocturnal hemoglobinuria: P. Hillmen et al., N. Engl. J. Med. 355, 1233 (2006).

Therapeutic Category

Anti-inflammatory.

Keywords

Anti-inflammatory (Biological Response Modifier)