6854. Opium

Nomenclature

Gum opium; crude opium.

Description and references

Air-dried latex from incised, unripe seed capsules of Papaver somniferum L., or P. album Mill., Papaveraceae. Constit. complex mixture of more than 20 alkaloids (20-30%) present as salts of meconic, lactic and sulfuric acids; volatile pyrazine derivatives responsible for the characteristic odor; meconin, sugars, proteins, gums, wax, fats, water. Morphine is the most important alkaloid and occurs to the extent of 10-16%, noscapine 4-8%, codeine 0.8-2.5%, papaverine 0.5-2.5%, thebaine 0.5-2%. For medicinal purposes, raw opium is dried at not above 70°, granulated or powdered, and adjusted with lactose or other inert diluent to contain 10-10.5% anhydr morphine. Historical review: M. J. Brownstein, Proc. Natl. Acad. Sci. USA 90, 5391-5393 (1993). Review of alkaloid extraction processes: R. J. Bryant, Chem. Ind. (London) 1988 (5), 146-153; of opium characterization methods: B. Remberg et al., Bull. Narc. 46, 79-108 (1994). Review of composition, pharmacology, and abuse: H. Kalant, Addiction 92, 267-277 (1997). HPLC analysis of alkaloid content: K. Yoshimatsu et al., Chem. Pharm. Bull. 53, 1446 (2005). Clinical use of opium tincture in neonatal abstinence syndrome: M. G. Coyle et al., J. Pediatr. 140, 561 (2002).

Properties

Pale olive-brown or gray, rounded, oval, brick-shaped or elongated, flattened masses with coarse surface, becoming hard or tough on storage. Internally, reddish brown and coarsely granular. Characteristic odor and very bitter taste.

Derivative

Deodorized opium.

Nomenclature

Denarcotized opium.

Properties

Powdered opium freed from its odor and nauseating substances by treatment with petr ether. Contains 10-10.5% anhydr morphine.

Derivative

Laudanum.

Nomenclature

Opium tincture.

Properties

Boiling water extract of opium mixed with dil alcohol. Contains 1 g anhydr morphine per 100 ml.

Derivative

Paregoric.

Nomenclature

Camphorated tincture of opium.

Properties

Mixture of powdered opium or opium tincture with benzoic acid, anise or other essential oil, glycerin, and alcohol. Contains 35-45 mg anhydr morphine per 100 ml.

Note

This is a controlled substance: 21 CFR, 1308.12.

Use

Largely for the manuf of morphine, codeine and other opium alkaloids.

Therapeutic Category

Analgesic; antidiarrheal.

Therapeutic Category (Veterinary)

Analgesic; antidiarrheal; antitussive.

Keywords

Analgesic; Opioids; Phenanthrenes; Antidiarrheal