Lidocaine is metabolized by CYP1A2 with some contribution from CYP3A4.
Metabolism
Enzyme: CYP1A2 [HSA:1544]; CYP3A4 [HSA:1576]
Interaction
Brite
USP drug classification [BR:br08302]
Anesthetics
Local Anesthetics
Lidocaine/ Tetracaine
D11553 Lidocaine and tetracaine
Drug groups [BR:br08330]
Metabolizing enzyme substrate
DG01892 CYP1A2 substrate
D11553 Lidocaine and tetracaine
DG01633 CYP3A/CYP3A4 substrate
DG02913 CYP3A4 substrate
D11553 Lidocaine and tetracaine
Drug metabolizing enzymes and transporters [br08309.html]
Drug metabolizing enzymes
D11553