Simeprevir


Entry
DG01246                     DGroup                                 
Name
Simeprevir
  Abbr
SMV
Type
Chemical
Member
D10081  
Simeprevir (JAN/USAN)
D10469  
Simeprevir sodium (JAN)
Class
Antiviral
 DG03198  Anti-HCV agent
  DG02001  HCV NS3/4A protease inhibitor
Metabolizing enzyme substrate
 DG01633  CYP3A/CYP3A4 substrate
Metabolizing enzyme inhibitor
 DG02852  CYP3A/CYP3A4 inhibitor
Transporter substrate
 DG01665  ABCB1 substrate
 DG02856  SLCO1B1 substrate
Transporter inhibitor
 DG01622  ABCB1 inhibitor
 DG02862  ABCG2 inhibitor
 DG02865  SLCO1B1 inhibitor
Remark
ATC code: J05AP05