Histamine receptor H1 antagonist


Entry
DG01482                     DGroup                                 
Name
Histamine receptor H1 antagonist
Type
Target
Member
DG00265  
Ketanserin
 D02363  
Ketanserin (USAN/INN)
 D08099  
Ketanserin tartrate
DG00381  
Thonzylamine
 D08587  
Thonzylamine (INN)
 D01801  
Thonzylamine hydrochloride (JAN/USAN)
DG00382  
Mepyramine
 D08183  
Mepyramine (INN)
 D05660  
Pyrilamine maleate (USP)
 D08184  
Mepyramine theophyllineacetate
DG00383  
Tripelennamine
 D08645  
Tripelennamine (INN)
 D02091  
Tripelennamine hydrochloride (USP)
 D06246  
Tripelennamine citrate
DG00384  
Chloropyramine
 D07195  
Chloropyramine (INN)
 D07679  
Chloropyramine hydrochloride
DG00385  
Promethazine
 D00494  
Promethazine (JAN/INN)
 D00480  
Promethazine hydrochloride (JP18/USP)  <JP/US>
 D01242  
Promethazine teoclate (JAN/INN)
 D03290  
Promethazine methylenedisalicylate (JAN)  <JP>
 D08432  
Promethazine maleate
 D08768  
Promethazine hibenzate  <JP>
DG00386  
Dimetindene
 D07853  
Dimetindene (INN)
 D01343  
Dimethindene maleate (USAN); Dimetindene maleate (JAN)
DG00387  
Clemastine
 D03535  
Clemastine (USAN)
 D00666  
Clemastine fumarate (JP18/USP)  <JP/US>
DG00388  
Bamipine
 D07197  
Bamipine (INN)
 D07492  
Bamipine dihydrochloride
 D07493  
Bamipine lactate
DG01100  
Pheniramine
 D08355  
Pheniramine (INN)
 D01174  
Pheniramine maleate (JAN/USP)
DG00389  
Isothipendyl
 D08091  
Isothipendyl (INN)
 D01143  
Isothipendyl hydrochloride (JAN)
DG00390  
Diphenhydramine
 D00300  
Diphenhydramine (JP18/INN)  <JP>
 D00669  
Diphenhydramine hydrochloride (JP18/USP)  <JP/US>
 D02419  
Diphenhydramine salicylate (JAN)
 D03285  
Diphenhydramine tannate (JP18)
 D03360  
Diphenhydramine laurylsulfate (JAN)  <JP>
 D03854  
Diphenhydramine citrate (USP)
 D00520  
Dimenhydrinate (JP18/USP/INN)  <JP/US>
DG00391  
Chlorphenoxamine
 D07198  
Chlorphenoxamine (INN)
 D07684  
Chlorphenoxamine hydrochloride
DG01035  
Levocabastine
 D08117  
Levocabastine (INN)
 D01717  
Levocabastine hydrochloride (JAN/USP)  <JP>
DG01036  
Azelastine
 D07483  
Azelastine (INN)
 D00659  
Azelastine hydrochloride (JP18/USP)  <JP/US>
DG01037  
Antazoline
 D07458  
Antazoline (INN)
 D02950  
Antazoline phosphate (USP)
 D07459  
Antazoline hydrochloride
DG01039  
Olopatadine
 D08293  
Olopatadine (INN)
 D01192  
Olopatadine hydrochloride (JP18/USP)  <JP/US>
D03166  
Bromodiphenhydramine hydrochloride (USP)
DG01094  
Diphenylpyraline
 D07862  
Diphenylpyraline (INN)
 D01172  
Diphenylpyraline hydrochloride (JAN)
 D01627  
Diphenylpyraline teoclate (JAN)
DG01095  
Carbinoxamine
 D07617  
Carbinoxamine (INN)
 D01336  
Carbinoxamine maleate (JAN/USP)  <US>
 D09808  
Carbinoxamine diphenyldisulfonate (JAN)
DG01096  
Doxylamine
 D07878  
Doxylamine (INN)
 D02327  
Doxylamine succinate (USP)
DG01097  
Brompheniramine
 D07543  
Brompheniramine (INN)
 D00663  
Brompheniramine maleate (USP)
DG01098  
Dexchlorpheniramine
 D07803  
Dexchlorpheniramine (INN)
 D00668  
Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18)  <JP/US>
DG01099  
Chlorphenamine
 D07398  
Chlorphenamine (INN)
 D00665  
Chlorpheniramine maleate (JP18/USP)  <JP>
 D03475  
Chlorpheniramine polistirex (USAN)
D03704  
Dexbrompheniramine maleate (USP)
DG01101  
Alimemazine
 D07125  
Alimemazine (INN); Trimeprazine (BAN)
 D02245  
Trimeprazine tartrate (USP); Alimemazine tartrate (JP18)  <JP>
D01324  
Mequitazine (JP18/INN)  <JP>
DG01104  
Buclizine
 D07547  
Buclizine (INN)
 D02089  
Buclizine hydrochloride (USAN)
DG01105  
Cyclizine
 D03621  
Cyclizine (INN)
 D02090  
Cyclizine lactate (BAN)
 D03622  
Cyclizine hydrochloride (USP)
DG01106  
Meclozine
 D08163  
Meclozine (BAN)
 D01317  
Meclizine hydrochloride (JAN/USP)  <US>
D01773  
Oxatomide (JAN/USAN/INN)  <JP>
DG01107  
Cetirizine
 D07662  
Cetirizine (INN)
 D00664  
Cetirizine hydrochloride (JP18/USP)  <JP/US>
DG01108  
Levocetirizine
 D07402  
Levocetirizine (USAN/INN)
 D08118  
Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN)  <JP/US>
DG01109  
Cyproheptadine
 D07765  
Cyproheptadine (INN)
 D02234  
Cyproheptadine hydrochloride (JP18/USP)  <JP/US>
DG01110  
Phenindamine
 D08353  
Phenindamine (INN)
 D02148  
Phenindamine tartrate (USAN)
DG01111  
Triprolidine
 D08648  
Triprolidine (INN)
 D01782  
Triprolidine hydrochloride (USP); Triprolidine hydrochloride hydrate (JAN)
DG01112  
Azatadine
 D07482  
Azatadine (INN)
 D00662  
Azatadine maleate (USP)
D00234  
Astemizole (JAN/USP/INN)
D00521  
Terfenadine (JAN/USAN/INN)
D00364  
Loratadine (JAN/USP/INN)  <JP/US>
DG01113  
Mebhydrolin
 D08161  
Mebhydrolin (INN)
 D01786  
Mebhydrolin napadisilate (JAN)
DG01114  
Deptropine
 D07404  
Deptropine (INN)
 D07790  
Deptropine citrate
DG01115  
Ketotifen
 D08105  
Ketotifen (INN)
 D01332  
Ketotifen fumarate (JP18/USAN)  <JP/US>
D02760  
Acrivastine (USAN/INN)
D01478  
Ebastine (JP18/USAN/INN)  <JP>
D07406  
Pimethixene (INN)
DG01116  
Epinastine
 D07900  
Epinastine (INN)
 D01713  
Epinastine hydrochloride (JAN)  <JP/US>
D01117  
Mizolastine (JAN/INN)
DG01117  
Fexofenadine
 D07958  
Fexofenadine (INN)
 D00671  
Fexofenadine hydrochloride (JP18/USP)  <JP/US>
D03693  
Desloratadine (JAN/USP/INN)  <JP/US>
DG01118  
Rupatadine
 D07407  
Rupatadine (INN)
 D08497  
Rupatadine fumarate (JAN)  <JP>
D09570  
Bilastine (JAN/INN)  <JP>
DG01144  
Emedastine
 D07890  
Emedastine (INN)
 D02249  
Emedastine difumarate (JP18/USP)  <JP>
D06552  
Alcaftadine (JAN/USAN/INN)  <US>
DG00843  
Dimetotiazine
 D07854  
Dimetotiazine (INN)
 D01902  
Fonazine mesylate (USAN); Dimetotiazine mesilate (JAN)  <JP>
DG00867  
Chlorpromazine
 D00270  
Chlorpromazine (USP/INN)
 D00789  
Chlorpromazine hydrochloride (JP18/USP)  <JP/US>
 D03274  
Chlorpromazine hibenzate (JAN)
 D04034  
Chlorpromazine phenolphthalinate (JAN)  <JP>
 D09819  
Chlorpromazine tannate (JAN)
DG00898  
Olanzapine
 D00454  
Olanzapine (JAN/USP/INN)  <JP/US>
 D06623  
Olanzapine pamoate (USAN)  <US>
DG00899  
Quetiapine
 D08456  
Quetiapine (INN)
 D00458  
Quetiapine fumarate (JP18/USP)  <JP/US>
DG00912  
Hydroxyzine
 D08054  
Hydroxyzine (INN)
 D00672  
Hydroxyzine hydrochloride (JP18/USP)  <JP/US>
 D01096  
Hydroxyzine pamoate (JP18/USP)  <JP/US>
DG00930  
Opipramol
 D08297  
Opipramol (INN)
 D01477  
Opipramol hydrochloride (JAN/USAN)
DG01005  
Cinnarizine
 D01295  
Cinnarizine (JAN/USAN/INN)
 D07734  
Cinnarizine dihydrochloride
DG01327  
Bepotastine
 D09705  
Bepotastine (USAN/INN)
 D01654  
Bepotastine besylate (USAN); Bepotastine besilate (JP18)  <JP/US>
DG01328  
Homochlorcyclizine
 D08041  
Homochlorcyclizine (INN)
 D01460  
Homochlorcyclizine hydrochloride (JP18)  <JP>
D04494  
Icotidine (USAN)
D05196  
Noberastine (USAN/INN)
D05742  
Rocastine hydrochloride (USAN)
D06021  
Tecastemizole (USAN/INN)
D06063  
Temelastine (USAN/INN)
D07860  
Dioxopromethazine hydrochloride
 » expand
Class
Anti-allergic agent
 DG01557  Histamine receptor antagonist