Grazoprevir


Entry
DG03051                     DGroup                                 
Name
Grazoprevir
  Abbr
GZR
Type
Chemical
Member
D11565  
Grazoprevir (USAN/INN)
D10639  
Grazoprevir (USAN); Grazoprevir hydrate (JAN)
Class
Antiviral
 DG03198  Anti-HCV agent
  DG02001  HCV NS3/4A protease inhibitor
Metabolizing enzyme substrate
 DG01633  CYP3A/CYP3A4 substrate
Metabolizing enzyme inhibitor
 DG02852  CYP3A/CYP3A4 inhibitor
Transporter substrate
 DG01665  ABCB1 substrate
 DG02856  SLCO1B1 substrate
Transporter inhibitor
 DG02862  ABCG2 inhibitor
Remark
ATC code: J05AP11