6842. Omalizumab

Nomenclature

CAS number: 242138-07-4
Anti-(human immunoglobulin E Fc region) immunoglobulin G (human-mouse monoclonal E25 clone pSVIE26 γ-chain) disulfide with human-mouse monoclonal E25 clone pSVIE26 κ-chain, dimer; olizumab; rhuMAb-E25; CGP-51901; Xolair (Novartis).

Description and references

Humanized monoclonal antibody directed against human immunoglobulin E (IgE). Complexes with circulating IgE to prevent the IgE-mediated degranulation of mast cells during an allergic reaction. Prepn: L. G. Presta et al., J. Immunol. 151, 2623 (1993). Pharmacokinetics and effect on circulating IgE levels in allergy patients: J. Corne et al., J. Clin. Invest. 99, 879 (1997). Clinical trial in allergic asthma: H. Milgrom et al., N. Engl. J. Med. 341, 1966 (1999); in allergic rhinitis: T. B. Casale et al., J. Am. Med. Assoc. 286, 2956 (2001). Reviews of clinical efficacy in allergic asthma: S. Holgate et al., Curr. Med. Res. Opin. 17, 233-240 (2001); G. D'Amato, Expert Opin. Biol. Ther. 3, 371-376 (2003).

Therapeutic Category

Antiallergic; antiasthmatic.

Keywords

Antiallergic; Antiasthmatic (Nonbronchodilator)