4063. Ferumoxides

Nomenclature

CAS number: 119683-68-0
AMI-25; Feridex (Advanced Magnetics); Endorem (Guerbet).

Description and references

Active ingredient of colloidal super paramagnetic iron oxide (SPIO) consisting of nonstoichiometric magnetite cores coated with dextran. Designed for use as hepatic MRI contrast agent. Prepn: E. V. Groman, L. Josephson, WO 8800060; eidem, US 4770183 (both 1988 to Advanced Magnetics). Pharmacokinetics: S. Majumdar et al., Invest. Radiol. 25, 771 (1990). Physical and chemical properties: C. W. Jung, P. Jacobs, Magn. Reson. Imaging 13, 661 (1995). Surface properties: C. W. Jung, ibid. 675. Clinical studies in hepatic imaging: T. J. Vogl et al., Radiology 198, 881 (1996); E. Senéterre et al., ibid. 200, 785 (1996). Series of articles on toxicology: Jpn. Pharmacol. Ther. 22, 57-141 (1994). Review of physicochemical characteristics and clinical applications: O. Clement et al., Top. Magn. Reson. Imaging 9, 167-182 (1998).

Properties

Aqueous suspension, black to reddish-brown liquid. Osmolality: ≈340 mOsm/kg. d 1.04.

Therapeutic Category

Diagnostic aid (MRI contrast agent).

Keywords

Diagnostic Aid (MRI Contrast Agent)