Nomenclature
CAS number: 54-28-4;
7616-22-0
(dl-form)
(2
R)-3,4-Dihydro-2,7,8-trimethyl-2-[(4
R,8
R)-4,8,12-trimethyltridecyl]-2
H-1-benzopyran-6-ol; (+)-2,7,8-trimethyl-2-(4,8,12-trimethyltridecyl)-6-chromanol; (
R,R,R)-γ-tocopherol; 7,8-dimethyltocol;
o-xylotocopherol.
C
28H
48O
2; mol wt 416.68.
C 80.71%, H 11.61%, O 7.68%.
Description and references
One of the naturally occurring forms of vitamin E, q.v. Most abundant tocopherol
in soybean and corn oils. Isoln by fractional crystn: Emerson et al., Science 83, 421 (1936); J. Biol. Chem. 113, 319 (1936); J. G. Baxter et al., J. Am. Chem. Soc. 65, 918 (1943).
Prepn of crystalline natural form: C. D. Robeson, J. Am. Chem. Soc. 65, 1660 (1943).
Comparison of bioactivity with α-tocopherol, q.v.: J. G. Bieri, R. P. Evarts, J. Nutr. 104, 850 (1974). Protective effects
vs reactive nitrogen oxide species: R. V. Cooney et al., Proc. Natl. Acad. Sci. USA 90, 1771 (1993); S. Christen et al., ibid. 94, 3217 (1997). HPLC determn in serum: A. Sobczak et al., J. Chromatogr. B 730, 265 (1999). Review of bioavailability, metabolism,
and activity: Q. Jiang et al., Am. J. Clin. Nutr. 74, 714-722 (2001).
Properties
Pale yellow, viscous oil. Has been crystallized
as transparent needles, mp 3
to 2°. bp0.1 200-210°. [α]546.125 2.4° (c = 8.59 in benzene); [α]546.125 +2.2° (c = 9.32 in ethanol). uv max: 298 nm
(E1%1cm 92.8). Insol in water. Freely
sol in oils, fats, acetone, alcohol, chloroform, ether, other fat
solvents. Very stable to heat and alkalies. Slowly oxidized by atmospheric
oxygen, rapidly by ferric and silver salts. Gradually darkens on
exposure to light.